Ranolazine

雷诺嗪

Report date: 2026/03/12 20:00:16
NMEFirst In Class

Base Information

Drug NameRanolazine
Drug Alias NameRanolazinum雷诺拉嗪雷诺嗓ranolazinaRanexa +[14
ClassificationSmall molecules > Heterocyclic drugs
Mechanisms of ActionSodium channel protein type V alpha subunit blockers
TargetsSodium channel protein type V alpha subunit
Therapy Area/IndicationsDiabetes Mellitus, Type 2Diabetes Mellitus, Type 1Myocardial Infarction +[26
Global Approved IndicationsAngina Pectoris
Approved Indications in ChinaN/A
Original Approved Country/TerritoryUnited States
Original Approved Date2006/01/27
Country/TerritoryCzechiaBelgiumCanada +[25
CombinationsNo
Global Highest StatusApproved
Highest Status in ChinaPhase 2 Clinical
Originator CompaniesGilead Sciences Inc
China Registration ClassN/A

Develop Information

Active IndicationsMyocardial InfarctionAngina, StableAngina Pectoris +[4
Inactive IndicationsDiabetes Mellitus, Type 2Diabetes Mellitus, Type 1Coronary Artery Disease +[22

Other Information

ATC CodeC01EB18