Grapiprant

N/A

Report date: 2026/03/12 20:00:16
NME

Base Information

Drug NameGrapiprant
Drug Alias NameRMX-1002AAT-007ARY-007CJ-023CJ-023,423 +[14
ClassificationSmall molecules > Heterocyclic drugs
Mechanisms of ActionProstanoid EP4 receptor antagonists
TargetsProstanoid EP4 receptor
Therapy Area/IndicationsSolid tumoursCancer PainPain +[10
Global Approved IndicationsN/A
Approved Indications in ChinaN/A
Original Approved Country/TerritoryN/A
Original Approved DateN/A
Country/TerritoryUnited StatesMainland China
CombinationsNo
Global Highest StatusPhase 2 Clinical
Highest Status in ChinaPhase 2 Clinical
China Registration ClassClass 1 Chemical Drug in China

Develop Information

Active IndicationsCancer PainPainColorectal Neoplasms
Inactive IndicationsSolid tumoursMastitisOsteoarthritis +[7

Other Information

ATC CodeN/A
Related LinksKEGG