Probenecid

丙磺舒

Report date: 2026/03/19 20:00:18
NME

Base Information

Drug NameProbenecid
Drug Alias Name璜舒Probenecidum黄舒羧苯磺丙胺羧苯磺胺 +[11
ClassificationSmall molecules > Heterocyclic drugs
Mechanisms of ActionCytochrome P450 2C9 inhibitorsOrganic Anion Transporter 3 inhibitorsUric acid transporter 1 inhibitors +[4
TargetsCytochrome P450 2C9Organic Anion Transporter 3Uric acid transporter 1 +[4
Therapy Area/IndicationsCoronavirus Disease 2019 (COVID-19)CravingAlcohol Abstinence +[10
Global Approved IndicationsHyperuricemiaGout
Approved Indications in ChinaGout
Original Approved Country/TerritoryUnited States
Original Approved Date1951/04/26
Country/TerritoryCanadaUnited StatesIndia +[4
CombinationsNo
Global Highest StatusApproved
Highest Status in ChinaApproved
Originator CompaniesMerck Sharp & Dohme Corp
China Registration ClassN/A

Develop Information

Active IndicationsCoronavirus Disease 2019 (COVID-19)CravingAlcohol Abstinence +[8
Inactive IndicationsHyperuricemiaHeart Failure, Systolic

Other Information

ATC CodeM04AB01